Palladium-catalyzed C2-acylation of indoles with aryl and alkyl aldehydes

Xiao Biao Yan; Yong Wen Shen; Dao Qian Chen; Pin Gao; Ying Xiu Li; Xian Rong Song; Xue Yuan Liu; Yong Min Liang

doi:10.1016/j.tet.2014.08.025

Palladium-catalyzed C2-acylation of indoles with aryl and alkyl aldehydes

Xiao Biao Yan
, Yong Wen Shen
, Dao Qian Chen
, Pin Gao
, Ying Xiu Li
, Xian Rong Song
, Xue Yuan Liu
, Yong Min Liang

Lanzhou University

Research output: Contribution to journal › Article › peer-review

39 Scopus citations

Abstract

A palladium-catalyzed C2-acylation of indoles with aryl and alkyl aldehydes via C-H functionalization is reported. The method shows excellent functional group tolerance and provides a straightforward way for the preparation of 2-aroylindoles.

Original language	English
Pages (from-to)	7490-7495
Number of pages	6
Journal	Tetrahedron
Volume	70
Issue number	41
DOIs	https://doi.org/10.1016/j.tet.2014.08.025
State	Published - 14 Oct 2014
Externally published	Yes

Keywords

2-Aroylindole
Acylation
Aldehyde
Indole
Palladium

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10.1016/j.tet.2014.08.025

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title = "Palladium-catalyzed C2-acylation of indoles with aryl and alkyl aldehydes",

abstract = "A palladium-catalyzed C2-acylation of indoles with aryl and alkyl aldehydes via C-H functionalization is reported. The method shows excellent functional group tolerance and provides a straightforward way for the preparation of 2-aroylindoles.",

keywords = "2-Aroylindole, Acylation, Aldehyde, Indole, Palladium",

author = "Yan, \{Xiao Biao\} and Shen, \{Yong Wen\} and Chen, \{Dao Qian\} and Pin Gao and Li, \{Ying Xiu\} and Song, \{Xian Rong\} and Liu, \{Xue Yuan\} and Liang, \{Yong Min\}",

year = "2014",

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day = "14",

doi = "10.1016/j.tet.2014.08.025",

language = "英语",

volume = "70",

pages = "7490--7495",

journal = "Tetrahedron",

issn = "0040-4020",

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TY - JOUR

T1 - Palladium-catalyzed C2-acylation of indoles with aryl and alkyl aldehydes

AU - Yan, Xiao Biao

AU - Shen, Yong Wen

AU - Chen, Dao Qian

AU - Gao, Pin

AU - Li, Ying Xiu

AU - Song, Xian Rong

AU - Liu, Xue Yuan

AU - Liang, Yong Min

PY - 2014/10/14

Y1 - 2014/10/14

N2 - A palladium-catalyzed C2-acylation of indoles with aryl and alkyl aldehydes via C-H functionalization is reported. The method shows excellent functional group tolerance and provides a straightforward way for the preparation of 2-aroylindoles.

AB - A palladium-catalyzed C2-acylation of indoles with aryl and alkyl aldehydes via C-H functionalization is reported. The method shows excellent functional group tolerance and provides a straightforward way for the preparation of 2-aroylindoles.

KW - 2-Aroylindole

KW - Acylation

KW - Aldehyde

KW - Indole

KW - Palladium

UR - https://www.scopus.com/pages/publications/84907086041

U2 - 10.1016/j.tet.2014.08.025

DO - 10.1016/j.tet.2014.08.025

M3 - 文章

AN - SCOPUS:84907086041

SN - 0040-4020

VL - 70

SP - 7490

EP - 7495

JO - Tetrahedron

JF - Tetrahedron

IS - 41

ER -

Palladium-catalyzed C2-acylation of indoles with aryl and alkyl aldehydes

Abstract

Keywords

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